SCHEMBL2245606

SCHEMBL2245606

NC(=O)[C@H](CCC(=O)O)NC(=O)c1ccc(-c2ccc(O)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 3/20 0.65
HPGDS O60760 4/20 0.65
CA1 P00915 3/20 0.56
CA12 O43570 1/20 0.56
CA9 Q16790 1/20 0.56
PTPN1 P18031 1/20 0.54
CA2 P00918 4/20 0.53
ADAMTS5 Q9UNA0 2/20 0.53
ADAMTS4 O75173 1/20 0.53
MMP2 P08253 2/20 0.47
MMP8 P22894 2/20 0.47
KDM4E B2RXH2 1/20 0.47
HPGD P15428 1/20 0.47
FOLH1 Q04609 2/20 0.46
NAALAD2 Q9Y3Q0 1/20 0.46
MMP13 P45452 1/20 0.46
DEGS1 O15121 1/20 0.46
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2245321 0.92 MMP12 (0.76) MMP12HPGDSCA1CA12CA9
SCHEMBL2246054 0.92 MMP12 (0.76) MMP12HPGDSCA1CA12CA9
SCHEMBL2249740 0.86 MMP12 (0.66) MMP12HPGDSCA1CA12CA9
SCHEMBL4622966 0.86 MMP12 (0.63) MMP12HPGDSCA1CA12CA9
SCHEMBL2249688 0.85 MMP12 (0.61) MMP12HPGDSCA1CA12CA9
SCHEMBL2246505 0.84 MMP12 (0.64) MMP12HPGDSCA1CA12CA9
SCHEMBL2246702 0.84 MMP12 (0.60) MMP12HPGDSCA1CA12CA9
SCHEMBL2247871 0.84 MMP12 (0.60) MMP12HPGDSCA1CA12CA9
SCHEMBL28108803 0.84 HPGDS (0.69) MMP12HPGDSCA1CA12CA9
SCHEMBL10518630 0.84 HPGDS (0.69) MMP12HPGDSCA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed