SCHEMBL2249688

SCHEMBL2249688

CCc1ccc(-c2ccc(C(=O)N[C@@H](CCC(=O)O)C(N)=O)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 3/20 0.61
CA1 P00915 3/20 0.58
CA12 O43570 2/20 0.58
CA9 Q16790 2/20 0.58
HPGDS O60760 3/20 0.55
PTPN1 P18031 1/20 0.54
ADAMTS5 Q9UNA0 2/20 0.53
ADAMTS4 O75173 1/20 0.53
MMP2 P08253 2/20 0.53
MMP8 P22894 2/20 0.53
TAS1R3 Q7RTX0 1/20 0.51
TAS1R1 Q7RTX1 1/20 0.51
CA2 P00918 3/20 0.50
MMP13 P45452 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
LMNA P02545 1/20 0.48
HSD17B10 Q99714 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4622966 0.88 MMP12 (0.63) MMP12CA1CA12CA9HPGDS
SCHEMBL2246054 0.88 MMP12 (0.76) MMP12CA1CA12CA9HPGDS
SCHEMBL2245321 0.88 MMP12 (0.76) MMP12CA1CA12CA9HPGDS
SCHEMBL403968 0.86 ADAMTS5 (0.58) MMP12CA1CA12CA9ADAMTS5
SCHEMBL2245606 0.85 MMP12 (0.65) MMP12CA1CA12CA9HPGDS
SCHEMBL2249692 0.85 CA2 (0.62) CA1CA12CA9MMP2TAS1R3
SCHEMBL2246912 0.84 MMP12 (0.58) MMP12CA1CA12CA9HPGDS
SCHEMBL27540278 0.84 TAS1R3 (0.68) CA1CA12CA9TAS1R3TAS1R1
SCHEMBL2246505 0.84 MMP12 (0.64) MMP12CA1CA12CA9HPGDS
SCHEMBL2249740 0.83 MMP12 (0.66) MMP12CA1CA12CA9HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed