SCHEMBL2249740

SCHEMBL2249740

NC(=O)[C@H](CCC(=O)O)NC(=O)c1ccc(-c2ccncc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 2/20 0.66
HPGDS O60760 3/20 0.56
CA1 P00915 2/20 0.54
CA12 O43570 1/20 0.54
CA9 Q16790 1/20 0.54
GSK3B P49841 8/20 0.53
ROCK1 Q13464 8/20 0.53
CLK4 Q9HAZ1 8/20 0.53
RPS6KA5 O75582 7/20 0.53
PRKG1 Q13976 7/20 0.53
PKN2 Q16513 7/20 0.53
GSK3A P49840 7/20 0.53
AKT1 P31749 6/20 0.53
PRKCD Q05655 6/20 0.53
PRKG2 Q13237 6/20 0.53
ROCK2 O75116 6/20 0.53
MAPK1 P28482 6/20 0.53
SGK2 Q9HBY8 6/20 0.53
MAP4K4 O95819 5/20 0.53
RPS6KB1 P23443 5/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2245321 0.89 MMP12 (0.76) MMP12HPGDSCA1CA12CA9
SCHEMBL2246054 0.89 MMP12 (0.76) MMP12HPGDSCA1CA12CA9
SCHEMBL2244000 0.88 MMP12 (0.61) MMP12HPGDSCA1CA12CA9
SCHEMBL2245606 0.86 MMP12 (0.65) MMP12HPGDSCA1CA12CA9
SCHEMBL4622966 0.84 MMP12 (0.63) MMP12HPGDSCA1CA12CA9
SCHEMBL2249747 0.84 CA2 (0.63) MMP12CA1GSK3BROCK1CLK4
SCHEMBL2249688 0.83 MMP12 (0.61) MMP12HPGDSCA1CA12CA9
SCHEMBL2246505 0.82 MMP12 (0.64) MMP12HPGDSCA1CA12CA9
SCHEMBL2246702 0.82 MMP12 (0.60) MMP12HPGDSCA1CA12CA9
SCHEMBL2247871 0.82 MMP12 (0.60) MMP12HPGDSCA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed