SCHEMBL22468348

SCHEMBL22468348

Nc1cnn(C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20523552 0.82 EPHX2 (0.30)
SCHEMBL19557881 0.76 MAPT (0.32) MAPTLMNAALDH1A1PKML3MBTL1
SCHEMBL20053912 0.76 MAPT (0.32) MAPTLMNAALDH1A1PKML3MBTL1
SCHEMBL10770145 0.76 LMNA (0.30) MAPTLMNA
SCHEMBL25047557 0.71 MPO (0.34)
SCHEMBL13129994 0.71 NOS1 (0.38) MAPTALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL30716649 0.70 GABRA1 (0.48)
SCHEMBL15652485 0.69 KIT (0.49) MAPTLMNAALDH1A1PKML3MBTL1
SCHEMBL23210319 0.69
SCHEMBL23229773 0.69 PDK2 (0.39) MAPTLMNAALDH1A1PKML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025038863-A1 INDOLE AND PYRROLOYPYRIDINE DERIVATIVES AS GPR17 MODULATORS BIOGEN MA INC. (US) 2025-02-20 WO disclosed
CN-118359634-A Pyrazole derivative and medical use thereof 正大天晴药业集团股份有限公司 2024-07-19 CN disclosed
US-20230365592-A1 COMPOUNDS AND METHODS USEFUL FOR STABILIZING PHENYLALANINE HYDROXYLASE MUTATIONS AGIOS PHARMACEUTICALS, INC. 2023-11-16 US disclosed
US-20230183217-A1 INHIBITORS OF LRRK2 KINASE HALIA THERAPEUTICS INC (US) 2023-06-15 US disclosed
US-11578061-B2 Inhibitors of LRRK2 kinase Halia Therapeutics, Inc. (US) 2023-02-14 US disclosed
EP-3941922-A1 INHIBITORS OF RAF KINASES Kinnate Biopharma Inc. (US) 2022-01-26 EP disclosed
CN-113874381-A Inhibitors of RAF kinase 金耐特生物制药公司 2021-12-31 CN disclosed
WO-2021147952-A1 PYRIMIDOPYRROLE COMPOUND 江苏先声药业有限公司 2021-07-29 WO disclosed
EP-3774782-A2 ATF6 INHIBITORS AND USES THEREOF Black Belt TX Ltd (GB) 2021-02-17 EP disclosed
WO-2020198058-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2020-10-01 WO disclosed
WO-2020198058-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2020-10-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230183217-A1 INHIBITORS OF LRRK2 KINASE LRRK2, SNCA, PRKAR2B MAPT 422/4885LMNA 532/4885ALDH1A1 2661/4885
US-20230365592-A1 COMPOUNDS AND METHODS USEFUL FOR STABILIZING PHENYLALANINE HYDROXYLASE MUTATIONS PAH, KDM8, PHF8 MAPT 2359/4885LMNA 798/4885ALDH1A1 865/4885
US-11578061-B2 Inhibitors of LRRK2 kinase LRRK2, SNCA, PRKAR2B MAPT 422/4885LMNA 532/4885ALDH1A1 2661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.