SCHEMBL22474477

SCHEMBL22474477

Fc1cccc2c1OC1CCC[C@@H](C2)Oc2c(F)cccc2C1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.38
DRD3 P35462 5/20 0.38
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
HTR1A P08908 3/20 0.33
HTR7 P34969 3/20 0.33
ADRA2A P08913 1/20 0.32
TERT O14746 1/20 0.31
PARP1 P09874 3/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22474530 1.00 DRD2 (0.38) DRD2DRD3PRKAB2PRKAG1PRKAA2
SCHEMBL22474523 0.93 DRD2 (0.40) DRD2DRD3PRKAB2PRKAG1PRKAA2
SCHEMBL22474522 0.82 PRKAB2 (0.36) DRD2DRD3PRKAB2PRKAG1PRKAA2
SCHEMBL22474545 0.81 PRKAB2 (0.35) DRD2DRD3PRKAB2PRKAG1PRKAA2
SCHEMBL22474535 0.79 HTR1A (0.33) HTR1AHTR7ADRA2APARP1
SCHEMBL22474507 0.79 TDP1 (0.36) HTR1AHTR7ADRA2APARP1
SCHEMBL22474494 0.79 PARP1 (0.31) PARP1
SCHEMBL22474487 0.79 HTR1A (0.33) HTR1AHTR7ADRA2APARP1
SCHEMBL22474526 0.79 DRD2 (0.42) DRD2DRD3
SCHEMBL22474552 0.78 PRKAB2 (0.34) DRD2DRD3PRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2876108-B1 COMPOUNDS OF CHIRAL AROMATIC SPIROKETAL DIPHOSPHINE LIGANDS, PREPARATION METHODS AND USES THEREOF SHANGHAI INST ORGANIC CHEMISTRY CAS (CN) 2020-09-30 EP disclosed