SCHEMBL22474535

SCHEMBL22474535

Brc1cccc2c1OC1CCC[C@H](C2)Oc2c(Br)cccc2C1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
HTR2B P41595 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
ADRA1A P35348 1/20 0.32
PARP1 P09874 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22474487 1.00 HTR1A (0.33) HTR1AHTR7HTR2BTMEM97SIGMAR1
SCHEMBL22474494 0.79 PARP1 (0.31) PARP1
SCHEMBL22474526 0.79 DRD2 (0.42)
SCHEMBL22474477 0.79 DRD2 (0.38) HTR1AHTR7ADRA2APARP1
SCHEMBL22474507 0.79 TDP1 (0.36) HTR1AHTR7HTR2BADRA2AADRA2B
SCHEMBL22474530 0.79 DRD2 (0.38) HTR1AHTR7ADRA2APARP1
SCHEMBL4596028 0.74 PARP1 (0.33) PARP1
SCHEMBL4596031 0.74 PARP1 (0.54) HTR1APARP1
SCHEMBL13993008 0.71 PRKAB2 (0.36) PARP1
SCHEMBL22474508 0.71 DRD1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2876108-B1 COMPOUNDS OF CHIRAL AROMATIC SPIROKETAL DIPHOSPHINE LIGANDS, PREPARATION METHODS AND USES THEREOF SHANGHAI INST ORGANIC CHEMISTRY CAS (CN) 2020-09-30 EP disclosed