SCHEMBL22476441

SCHEMBL22476441

COC(C(C)C(=O)NC(Cc1ccccc1)/C(N)=N/NN)C1CCCN1C=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
GAA P10253 1/20 0.36
MMP1 P03956 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.36
THRB P10828 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
F2 P00734 1/20 0.35
PRSS1 P07477 1/20 0.35
IL2RA P01589 1/20 0.35
ALB P02768 1/20 0.35
IL2 P60568 1/20 0.35
PSMB8 P28062 2/20 0.35
PSMB5 P28074 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25949990 0.88 ACE (0.46) ACEGAAALDH1A1THRBCYP2C9
SCHEMBL23154537 0.88 ACE (0.46) ACEGAAALDH1A1THRBCYP2C9
SCHEMBL18688556 0.88 ACE (0.46) ACEGAAALDH1A1THRBCYP2C9
SCHEMBL22476506 0.87 ACE (0.41) ACEOPRM1OPRD1OPRK1GAA
SCHEMBL21699258 0.87 CYP2C9 (0.49) GAAATML3MBTL1ALDH1A1THRB
SCHEMBL21699268 0.87 CYP2C9 (0.49) GAAATML3MBTL1ALDH1A1THRB
SCHEMBL19443278 0.86 MMP1 (0.44) ACEGAAMMP1ALDH1A1THRB
SCHEMBL22476544 0.86 MMP1 (0.44) ACEMMP1
SCHEMBL18683750 0.84 NPC1 (0.41) GAAATML3MBTL1ALDH1A1
SCHEMBL22476529 0.83 L3MBTL1 (0.45) ACEGAAMMP1ATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3303366-B1 DERIVATIVES OF DOLASTATIN 10 AND USES THEREOF NEWBIO THERAPEUTICS INC (CN) 2020-09-30 EP disclosed