SCHEMBL2248588

SCHEMBL2248588

NC(=O)[C@H](CCC(=O)O)NC(=O)c1ccc(-c2ccc(OCc3ccc4ccccc4c3)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 2/20 0.57
PTPN1 P18031 3/20 0.56
DHFR P00374 3/20 0.54
HPGDS O60760 2/20 0.52
NPC1 O15118 1/20 0.51
MAPT P10636 1/20 0.51
CTSL P07711 1/20 0.49
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
CTSK P43235 1/20 0.49
PLA2G4B P0C869 1/20 0.49
FFAR1 O14842 2/20 0.48
AKR1B1 P15121 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47
MMP13 P45452 2/20 0.47
ADAMTS4 O75173 1/20 0.47
MMP2 P08253 1/20 0.46
MMP8 P22894 1/20 0.46
CA2 P00918 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2247647 0.90 MMP12 (0.62) MMP12PTPN1DHFRHPGDSFFAR1
SCHEMBL2251669 0.90 MMP12 (0.61) MMP12PTPN1DHFRHPGDSMAPT
SCHEMBL2248592 0.88 DHFR (0.54) PTPN1DHFRNPC1MAPTCTSL
SCHEMBL3584792 0.87 FOLH1 (0.54) MMP12DHFRCTSLCTSBCTSS
SCHEMBL2249553 0.86 MMP12 (0.67) MMP12PTPN1HPGDSCTSLCTSB
SCHEMBL2247420 0.85 MMP12 (0.56) MMP12PTPN1DHFRHPGDSNPC1
SCHEMBL2246953 0.85 GRM5 (0.57) MMP12PTPN1DHFRHPGDSMMP13
SCHEMBL2245261 0.85 MMP12 (0.56) MMP12PTPN1DHFRHPGDSNPC1
SCHEMBL2243988 0.83 MMP12 (0.53) MMP12PTPN1DHFRHPGDSMAPT
SCHEMBL2250713 0.83 MMP12 (0.54) MMP12DHFRHPGDSNPC1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed