SCHEMBL22476478

SCHEMBL22476478

COCCOCCOCCNC(=O)C(Cc1ccccc1)NC(=O)C(C)C(OC)C1CCCN1C=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 5/20 0.42
TACR2 P21452 5/20 0.38
ACE P12821 2/20 0.37
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRND Q07001 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
AKT1 P31749 1/20 0.36
MMP1 P03956 1/20 0.36
FCER2 P06734 1/20 0.36
CPA1 P15085 1/20 0.35
CPA2 P48052 1/20 0.35
CPA4 Q9UI42 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22476529 0.89 L3MBTL1 (0.45) TACR2ACEL3MBTL1AKT1MMP1
SCHEMBL22476544 0.86 MMP1 (0.44) ACEMMP1FCER2
SCHEMBL19443278 0.86 MMP1 (0.44) ACEMMP1FCER2
SCHEMBL23154537 0.86 ACE (0.46) ACECPA1
SCHEMBL18688556 0.86 ACE (0.46) ACECPA1
SCHEMBL25949990 0.86 ACE (0.46) ACECPA1
SCHEMBL22476555 0.85 TACR2 (0.40) CAPN1TACR2ACE
SCHEMBL22476506 0.85 ACE (0.41) ACEL3MBTL1
SCHEMBL21699268 0.85 CYP2C9 (0.49) L3MBTL1
SCHEMBL21699258 0.85 CYP2C9 (0.49) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3303366-B1 DERIVATIVES OF DOLASTATIN 10 AND USES THEREOF NEWBIO THERAPEUTICS INC (CN) 2020-09-30 EP disclosed