SCHEMBL22483009

SCHEMBL22483009

C/C=N\c1c(NC)c(=O)n(CCNC(=O)CCC)c(=O)n1C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP2 P42575 1/20 0.35
GPR84 Q9NQS5 1/20 0.34
TP53 P04637 2/20 0.34
THRB P10828 2/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
ADORA1 P30542 3/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22483005 0.91 TP53 (0.34) TP53THRBPOLBL3MBTL1MTNR1A
SCHEMBL22483038 0.79 ALDH1A1 (0.40) ALDH1A1
SCHEMBL22483004 0.76 GAA (0.47) POLBALDH1A1NPSR1
SCHEMBL13413721 0.71 CASP2 (0.50) CASP2THRBPOLBL3MBTL1MTNR1A
SCHEMBL9772333 0.62 TSHR (0.48) CASP2TP53MTNR1AMTNR1BALDH1A1
SCHEMBL22521716 0.61 TOP2A (0.41) ALDH1A1
SCHEMBL7537764 0.59 CASP2 (0.86) CASP2
SCHEMBL16120761 0.59 PTGS1 (0.46) CASP2MTNR1AMTNR1BALDH1A1TSHR
SCHEMBL2633147 0.58 CASP2 (0.70) CASP2ALDH1A1
SCHEMBL13413716 0.58 MEN1 (0.52) TP53THRBPOLBL3MBTL1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020192665-A1 NUCLEOSIDE DERIVATIVE FOR PREVENTING AND TREATING INFLAMMATION AND APPLICATION THEREOF 四川大学华西医院 2020-10-01 WO disclosed