SCHEMBL22493023

SCHEMBL22493023

CCOC(=O)c1cn(-c2ccccc2[N+](=O)[O-])nc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.45
ALDH1A1 P00352 3/20 0.45
GAA P10253 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
DGAT1 O75907 7/20 0.45
SLC5A1 P13866 1/20 0.44
SLC5A2 P31639 1/20 0.44
POLB P06746 1/20 0.43
MAPK1 P28482 2/20 0.41
NPC1 O15118 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
CES2 O00748 1/20 0.40
ACHE P22303 1/20 0.40
CES1 P23141 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL407653 0.84 DGAT1 (0.49) MAPTALDH1A1GAASMN1; SMN2DGAT1
SCHEMBL407225 0.83 DGAT1 (0.48) MAPTALDH1A1SMN1; SMN2DGAT1POLB
SCHEMBL442691 0.83 DGAT1 (0.61) ALDH1A1GAASMN1; SMN2DGAT1MAPK1
SCHEMBL408707 0.82 PDE4B (0.50) ALDH1A1DGAT1MAPK1NPSR1
SCHEMBL407661 0.81 DGAT1 (0.47) MAPTALDH1A1GAADGAT1MAPK1
SCHEMBL22493020 0.81 MAPT (0.62) MAPTALDH1A1SMN1; SMN2DGAT1MAPK1
SCHEMBL408172 0.79 NPSR1 (0.60) MAPTALDH1A1SMN1; SMN2DGAT1POLB
SCHEMBL408667 0.77 DGAT1 (0.43) ALDH1A1GAADGAT1MAPK1LMNA
SCHEMBL20304409 0.76 TDP1 (0.46) SMN1; SMN2DGAT1MAPK1NPC1NFKB1
SCHEMBL407666 0.76 DGAT1 (0.62) MAPTALDH1A1GAASMN1; SMN2DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11655203-B2 Nitration ETH ZURICH (CH) 2023-05-23 US disclosed
US-20220009875-A1 NITRATION ETH ZURICH (CH) 2022-01-13 US disclosed
CN-113302186-A Nitration 瑞士苏黎世联邦理工学院 2021-08-24 CN disclosed
EP-3717464-B1 NITRATION ETH ZUERICH (CH) 2021-06-16 EP disclosed
EP-3717464-A1 NITRATION ETH Zurich (CH) 2020-10-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220009875-A1 NITRATION NOS1, NOS2, NOS3 MAPT 3137/4885ALDH1A1 2335/4885GAA 4180/4885
US-11655203-B2 Nitration NOS1, NOS2, NOS3 MAPT 3137/4885ALDH1A1 2335/4885GAA 4180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.