SCHEMBL22497553

SCHEMBL22497553

O=C(Nc1ccccc1C(=O)O)OCc1cc(F)cc(F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.52
NPC1 O15118 2/20 0.52
KDM4E B2RXH2 2/20 0.50
MGLL Q99685 2/20 0.50
GAA P10253 1/20 0.50
STAT1 P42224 1/20 0.50
HCAR2 Q8TDS4 2/20 0.48
LMNA P02545 1/20 0.47
CFD P00746 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CASP3 P42574 1/20 0.46
POLB P06746 1/20 0.46
PKM P14618 1/20 0.46
CTSV O60911 1/20 0.45
CTSL P07711 1/20 0.45
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MMP12 P39900 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22497489 0.87 KDM4E (0.61) RAB9ANPC1KDM4EMGLLHCAR2
SCHEMBL2233522 0.85 NPC1 (0.69) RAB9ANPC1KDM4EMGLLLMNA
SCHEMBL26030821 0.81 CASP3 (0.62) RAB9ANPC1KDM4EMGLLGAA
SCHEMBL5055502 0.80 NPC1 (0.58) RAB9ANPC1MGLLHCAR2CFD
SCHEMBL7122137 0.80 MGLL (0.65) RAB9ANPC1MGLLMEN1KMT2A
SCHEMBL22497537 0.78 TRPV1 (0.58) RAB9ANPC1MGLLMEN1KMT2A
SCHEMBL22497529 0.78 GRIK1 (0.59) RAB9ANPC1MGLLGAAMEN1
SCHEMBL30279458 0.78 GRIK1 (0.59) RAB9ANPC1MGLLGAAMEN1
SCHEMBL10489819 0.76 KMT2A (0.63) RAB9ANPC1KDM4EGAALMNA
SCHEMBL8115672 0.76 ALDH1A1 (0.63) RAB9ANPC1KDM4EMGLLLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020199945-A1 ORTHO-CARBONYL AMINO-SUBSTITUTED BENZENE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国医学科学院药物研究所 2020-10-08 WO disclosed
WO-2020199945-A1 ORTHO-CARBONYL AMINO-SUBSTITUTED BENZENE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国医学科学院药物研究所 2020-10-08 WO disclosed