SCHEMBL2249769

SCHEMBL2249769

CC(O)C(=O)N1CCC(N)C1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 16/20 0.45
DPP8 Q6V1X1 6/20 0.45
DPP9 Q86TI2 3/20 0.45
DPP7 Q9UHL4 8/20 0.41
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
KCNH2 Q12809 1/20 0.37
GNAI3 P08754 1/20 0.37
GNAO1 P09471 1/20 0.37
GNAI1 P63096 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2249766 1.00 DPP4 (0.45) DPP4DPP8DPP9DPP7MEN1
SCHEMBL20385048 1.00 DPP4 (0.45) DPP4DPP8DPP9DPP7MEN1
SCHEMBL3397414 1.00 DPP4 (0.45) DPP4DPP8DPP9DPP7MEN1
SCHEMBL3424335 1.00 DPP4 (0.45) DPP4DPP8DPP9DPP7MEN1
SCHEMBL3400585 0.89 TLR9 (0.37) DPP4DPP8DPP9DPP7MEN1
SCHEMBL3399856 0.89 TLR9 (0.37) DPP4DPP8DPP9DPP7MEN1
SCHEMBL985368 0.88 MEN1 (0.46) DPP4DPP8DPP9DPP7MEN1
SCHEMBL985369 0.88 MEN1 (0.46) DPP4DPP8DPP9DPP7MEN1
SCHEMBL5396145 0.86 DPP4 (0.46) DPP4DPP8DPP9DPP7MEN1
SCHEMBL12414282 0.86 DPP4 (0.46) DPP4DPP8DPP9DPP7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8759535-B2 Substituted fused imidazole derivatives, pharmaceutical compositions, and methods of use thereof HIGH POINT PHARMACEUTICALS, LLC (US) 2014-06-24 US disclosed
US-20110201604-A1 Substituted Fused Imidazole Derivatives, Pharmaceutical Compositions, and Methods of Use Thereof HIGH POINT PHARMACEUTICALS, LLC (US) 2011-08-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110201604-A1 Substituted Fused Imidazole Derivatives, Pharmaceutical Compositions, and Methods of Use Thereof HMOX2, HMOX1, PTGS2 DPP4 502/4885DPP8 213/4885DPP9 354/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.