SCHEMBL22498698

SCHEMBL22498698

CC(=CCc1c(O)cc(O)c2c1OC(c1ccc(O)cc1)C(=O)C2)CCC(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 4/20 0.49
ESR1 P03372 6/20 0.46
ESR2 Q92731 4/20 0.46
CACNA1H O95180 3/20 0.46
AKR1B10 O60218 2/20 0.46
AKR1B1 P15121 2/20 0.46
CACNA1G O43497 2/20 0.46
MAOA P21397 1/20 0.46
PDE5A O76074 1/20 0.46
ACHE P22303 2/20 0.42
PTGS2 P35354 2/20 0.42
TP53 P04637 1/20 0.42
MDM2 Q00987 1/20 0.42
CYP19A1 P11511 1/20 0.41
ELANE P08246 3/20 0.41
PDPK1 O15530 1/20 0.40
PRKCA P17252 1/20 0.40
BACE1 P56817 1/20 0.40
PRKCQ Q04759 1/20 0.40
PTPN1 P18031 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3368570 0.87 ESR1 (0.59) ABCG2ESR1ESR2CACNA1HAKR1B10
SCHEMBL5430100 0.80 ESR1 (0.43) ABCG2ESR1ESR2CACNA1HAKR1B10
SCHEMBL22498697 0.79 ABCG2 (0.78) ABCG2ESR1ESR2CACNA1HAKR1B10
SCHEMBL29379960 0.79 ABCG2 (0.78) ABCG2ESR1ESR2CACNA1HAKR1B10
SCHEMBL4758125 0.73 ESR2 (0.39) ESR1ESR2AKR1B1PTGS2CYP19A1
SCHEMBL19221566 0.71 ABCG2 (0.75) ABCG2ESR1ESR2CACNA1HAKR1B10
SCHEMBL27950799 0.70 TAS2R31 (0.39) ESR1ESR2CYP19A1PTPN1MAPT
Sophoraflavanone A SCHEMBL29624617 0.66 ABCG2 (1.00) ABCG2ESR1ESR2CACNA1HAKR1B10
Sophoraflavanone A SCHEMBL141996 0.66 ABCG2 (1.00) ABCG2ESR1ESR2CACNA1HAKR1B10
SCHEMBL349722 0.64 CYP3A4 (0.52) ESR1ESR2AKR1B1PTGS2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220128556-A1 METHODS OF DIAGNOSING DISEASE 4D Pharma Cork Limited (IE) 2022-04-28 US disclosed
CN-114040986-A Method of diagnosing disease 4D制药科克有限公司 2022-02-11 CN disclosed
EP-3947743-A1 METHODS OF DIAGNOSING DISEASE 4D Pharma Cork Limited (IE) 2022-02-09 EP disclosed
WO-2020201457-A1 METHODS OF DIAGNOSING DISEASE 4D Pharma Cork Limited (IE) 2020-10-08 WO disclosed