SCHEMBL5430100

SCHEMBL5430100

C=CCc1c(O)cc(O)c2c1OC(c1ccc(O)cc1)C(=O)C2

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 12/20 0.43
ESR2 Q92731 11/20 0.43
ABCG2 Q9UNQ0 2/20 0.43
AKR1B10 O60218 2/20 0.43
AKR1B1 P15121 2/20 0.43
CACNA1H O95180 2/20 0.43
CACNA1G O43497 1/20 0.43
MAOA P21397 1/20 0.43
PDE5A O76074 1/20 0.43
CYP19A1 P11511 1/20 0.41
PDPK1 O15530 1/20 0.37
PRKCA P17252 1/20 0.37
BACE1 P56817 1/20 0.37
PRKCQ Q04759 1/20 0.37
PTPN1 P18031 1/20 0.36
SLC22A12 Q96S37 3/20 0.36
SLC2A9 Q9NRM0 2/20 0.36
XDH P47989 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3368570 0.86 ESR1 (0.59) ESR1ESR2ABCG2AKR1B10AKR1B1
SCHEMBL28635981 0.82 SLC22A12 (0.41) ESR1ESR2ABCG2AKR1B10AKR1B1
SCHEMBL22498698 0.80 ABCG2 (0.49) ESR1ESR2ABCG2AKR1B10AKR1B1
SCHEMBL4758125 0.80 ESR2 (0.39) ESR1ESR2AKR1B1CYP19A1XDH
SCHEMBL27950799 0.75 TAS2R31 (0.39) ESR1ESR2CYP19A1PTPN1
SCHEMBL2687105 0.73 ESR1 (0.76) ESR1ESR2ABCG2AKR1B10AKR1B1
SCHEMBL349722 0.71 CYP3A4 (0.52) ESR1ESR2AKR1B1CYP19A1BACE1
SCHEMBL3487578 0.71 CYP3A4 (0.52) ESR1ESR2AKR1B1CYP19A1BACE1
SCHEMBL19221566 0.69 ABCG2 (0.75) ESR1ESR2ABCG2AKR1B10AKR1B1
SCHEMBL5421506 0.68 CYP19A1 (0.38) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007053915-A2 NARINGENIN DERIVATIVES WITH SELECTIVITY ON ERS UNIVERSITEIT GENT (BE) 2007-05-18 WO disclosed