SCHEMBL22523908

SCHEMBL22523908

CCSN1CCC(c2cncc(Br)c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
L3MBTL4 Q8NA19 1/20 0.36
L3MBTL3 Q96JM7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ATM Q13315 1/20 0.36
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
GAA P10253 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD17B10 Q99714 1/20 0.34
CYP11B2 P19099 1/20 0.33
CACNA1I Q9P0X4 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21965642 0.85 DRD2 (0.41) CHRNB2CHRNA4L3MBTL4L3MBTL3L3MBTL1
SCHEMBL16271578 0.78 CYP11B2 (0.48) CHRNB2CHRNA4ATMGAAALDH1A1
SCHEMBL1426303 0.77 POLB (0.38) CHRNB2CHRNA4CYP11B2
SCHEMBL29845299 0.77 POLB (0.38) CHRNB2CHRNA4CYP11B2
SCHEMBL21965640 0.76 CHRNB2 (0.37) CHRNB2CHRNA4L3MBTL4L3MBTL3L3MBTL1
SCHEMBL16271594 0.76 ATM (0.52) L3MBTL4L3MBTL3L3MBTL1ATMGAA
SCHEMBL14991864 0.73 QDPR (0.51) L3MBTL4L3MBTL3L3MBTL1ATMGAA
SCHEMBL17581673 0.73 IDO1 (0.44) CHRNB2CHRNA4CYP11B2
SCHEMBL31014511 0.73 CYP11B2 (0.46) CHRNB2CHRNA4L3MBTL4L3MBTL3L3MBTL1
SCHEMBL16271599 0.69 DRD2 (0.41) CHRNB2CHRNA4L3MBTL4L3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3719019-B1 NEW 3,4-DIHYDRO-2H-ISOQUINOLINE-1-ONE AND 2,3-DIHYDRO-ISOINDOL-1-ONE COMPOUNDS HOFFMANN LA ROCHE (CH) 2022-01-19 EP disclosed
EP-3719019-A1 NEW 3,4-DIHYDRO-2H-ISOQUINOLINE-1-ONE AND 2,3-DIHYDRO-ISOINDOL-1-ONE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2020-10-07 EP disclosed