SCHEMBL22557500

SCHEMBL22557500

NC(=O)Oc1ccc(N)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
NNMT P40261 3/20 0.42
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
POLB P06746 2/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 2/20 0.40
KEAP1 Q14145 1/20 0.40
BRCA1 P38398 1/20 0.40
HBB P68871 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249721 0.84 KDM4E (0.44) KDM4EMEN1KMT2ANNMTADRA2A
SCHEMBL22557537 0.82 KDM4E (0.44) KDM4EMEN1KMT2ANNMTADRA2A
SCHEMBL29078226 0.80 NNMT (0.42) KDM4EMEN1KMT2ANNMTALDH1A1
SCHEMBL9572467 0.80 KMT2A (0.45) KDM4EMEN1KMT2ANNMTALDH1A1
SCHEMBL9018039 0.79 KDM4E (0.44) KDM4EMEN1KMT2ANNMTPOLB
SCHEMBL20639594 0.78 NNMT (0.41) KDM4EMEN1KMT2ANNMTALDH1A1
SCHEMBL28938017 0.78 ADRA2A (0.43) NNMTADRA2AADRA2BADRA2C
SCHEMBL2899777 0.78 KDM4E (0.46) KDM4EMEN1KMT2ANNMTADRA2A
SCHEMBL28476110 0.78 KDM4E (0.58) KDM4EMEN1KMT2ANNMTADRA2A
SCHEMBL22557367 0.78 KDM4E (0.41) KDM4EMEN1KMT2ANNMTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024131893-A1 IRE1α SMALL MOLECULE INHIBITORS SHANGHAI YI ZHONG XING BIOTECHNOLOGY CO., LTD. (CN) 2024-06-27 WO disclosed
CN-109562111-B CK2 inhibitors, compositions and methods thereof 北极星药业股份有限公司 2023-04-04 CN disclosed
EP-3956322-A1 JAK1 SELECTIVE KINASE INHIBITOR DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2022-02-23 EP disclosed
WO-2020211839-A1 JAK1 SELECTIVE KINASE INHIBITOR DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2020-10-22 WO disclosed