SCHEMBL22562387

SCHEMBL22562387

Cc1cccc(-c2cc(-n3c4ccc(-c5cccc(C#N)c5)cc4c4cc(-c5cccc(C#N)c5)ccc43)c(C#N)c(-n3c4ccc(-c5cccc(C#N)c5)cc4c4cc(-c5cccc(C#N)c5)ccc43)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 5/20 0.39
ADORA2A P29274 3/20 0.39
ADORA1 P30542 3/20 0.39
ADORA2B P29275 2/20 0.39
GRM5 P41594 1/20 0.39
ALDH1A3 P47895 1/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CLK4 Q9HAZ1 2/20 0.38
MAP4K4 O95819 1/20 0.37
GRM2 Q14416 1/20 0.37
WNT3A P56704 1/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
KMT2A Q03164 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562384 0.96 ADORA2A (0.39) TGFBR1ADORA2AADORA1ADORA2BGRM5
SCHEMBL23296383 0.91 TGFBR1 (0.40) TGFBR1ADORA2AADORA1ALDH1A1KMT2A
SCHEMBL21546805 0.86 ALDH1A3 (0.46) ADORA2AADORA1ADORA2BALDH1A3ALDH1A1
SCHEMBL23296293 0.85 IRAK4 (0.37) TGFBR1ADORA2AADORA1HIF1A
SCHEMBL22562313 0.85 METAP2 (0.37) TGFBR1
SCHEMBL22562197 0.85 TGFBR1 (0.37) TGFBR1ALDH1A1
SCHEMBL21547025 0.85 MAP4K4 (0.43) ADORA2AADORA1ADORA2BALDH1A3ALDH1A1
SCHEMBL22562530 0.83 ALDH1A3 (0.41) ADORA2AADORA1ADORA2BGRM5ALDH1A3
SCHEMBL21546828 0.83 CYP1A2 (0.39) ADORA2AADORA1ADORA2BGRM5ALDH1A3
SCHEMBL21546834 0.83 GRIA2 (0.39) ADORA2AADORA1ADORA2BALDH1A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3418278-B1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2020-10-21 EP disclosed