SCHEMBL22562822

SCHEMBL22562822

CCC(CC)n1nc[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
PDE9A O76083 2/20 0.33
PDE1C Q14123 1/20 0.33
PDE4A P27815 2/20 0.31
ADORA2A P29274 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
PDE4D Q08499 2/20 0.31
HCAR3 P49019 1/20 0.30
ACHE P22303 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8228728 0.78
SCHEMBL21211664 0.76 GAA (0.39) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8463363 0.64
SCHEMBL20644426 0.64 MAPT (0.33) CYP1A2PDE9APDE1CPDE4AADORA2A
SCHEMBL27762431 0.61 PDE4B (0.34) CYP1A2PDE4B
SCHEMBL2826206 0.60 ADORA2B (0.44) CYP1A2PDE4AADORA2APDE4BPDE4C
SCHEMBL910645 0.60
SCHEMBL16285366 0.59 MGLL (0.44) CYP1A2
SCHEMBL31330327 0.58 ADORA2A (0.33) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL31330241 0.58 ADORA2A (0.33) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3397629-B1 METALLOENZYME INHIBITOR COMPOUNDS NQP 1598 LTD (KY) 2023-04-19 EP claimed
WO-2024249959-A1 COMPOSITIONS REDUCING THE EXPRESSION OR ACTIVITY OF C1 GALT1 FOR TREATING EWING SARCOMA UNIVERSITY OF MASSACHUSETTS MEDICAL SCHOOL (US) 2024-12-05 WO disclosed
EP-3397629-B1 METALLOENZYME INHIBITOR COMPOUNDS NQP 1598 LTD (KY) 2023-04-19 EP disclosed
EP-3414216-B1 ARYLATION OF ALIPHATIC AMINES AAA CHEMISTRY APS (DK) 2020-10-21 EP disclosed