SCHEMBL22563092

SCHEMBL22563092

CCCC(CCC)c1ccc(C(=O)NC(=N)c2ccc(Nc3ccccc3F)cc2)nc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 3/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
AURKA O14965 3/20 0.38
NPC1 O15118 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HDAC1 Q13547 8/20 0.37
HDAC3 O15379 7/20 0.37
HDAC8 Q9BY41 3/20 0.37
HDAC2 Q92769 4/20 0.36
NCOR2 Q9Y618 4/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
DGAT1 O75907 1/20 0.35
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22563043 0.73 ALDH1A1 (0.35) MEN1KMT2ANPC1SMN1; SMN2HDAC1
SCHEMBL6717442 0.65 KDM4E (0.54) P4HTMMEN1KMT2A
SCHEMBL28537077 0.65 SMN1; SMN2 (0.50) P4HTMMEN1KMT2ANPC1SMN1; SMN2
SCHEMBL25605312 0.64 PRKAB2 (0.43) NPC1SMN1; SMN2RAB9A
SCHEMBL22563017 0.63 HDAC1 (0.37) HDAC1HDAC3HDAC2NCOR2HDAC6
SCHEMBL27308949 0.60 TAS1R3 (0.39) MEN1KMT2ASMN1; SMN2TAS1R3TAS1R1
SCHEMBL30763190 0.60 SMN1; SMN2 (0.60) P4HTMMEN1KMT2ANPC1SMN1; SMN2
SCHEMBL21595582 0.60 SMN1; SMN2 (0.60) P4HTMMEN1KMT2ANPC1SMN1; SMN2
SCHEMBL22116941 0.59 GAA (0.50) MEN1KMT2AAURKANPC1SMN1; SMN2
SCHEMBL20178617 0.58 KDM4E (0.54) P4HTMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed