SCHEMBL22563043

SCHEMBL22563043

CCCCC(CCC)c1ccc(C(=O)NC(=N)c2ccc(Nc3ccccc3P)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HDAC1 Q13547 4/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
HDAC3 O15379 2/20 0.34
HDAC2 Q92769 2/20 0.34
BDKRB2 P30411 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
S1PR3 Q99500 2/20 0.32
S1PR4 O95977 1/20 0.31
POLB P06746 1/20 0.31
BLM P54132 1/20 0.31
PRSS1 P07477 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562998 0.86 MAPK14 (0.33) HDAC1HDAC3HDAC2PLK1PLK3
SCHEMBL22563014 0.81 MAPK1 (0.34) MAPK1HDAC1PRSS1
SCHEMBL22563092 0.73 P4HTM (0.41) MEN1KMT2ASMN1; SMN2HDAC1HDAC8
SCHEMBL22562963 0.68 MAPK14 (0.39) ALDH1A1MEN1MAPTKMT2AHDAC1
SCHEMBL28533240 0.67 BDKRB2 (0.49) ALDH1A1MAPK1HDAC8HDAC6BDKRB2
SCHEMBL22563037 0.66 RARB (0.47) ALDH1A1MEN1MAPTKMT2A
SCHEMBL8760481 0.64 ALDH1A1 (0.50) ALDH1A1MEN1MAPTMAPK1KMT2A
SCHEMBL11960754 0.63 DEGS1 (0.51) MEN1KMT2AHDAC1HDAC8HDAC6
SCHEMBL8759863 0.63 NR1I2 (0.47) ALDH1A1MEN1MAPTMAPK1KMT2A
SCHEMBL21164999 0.62 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed