SCHEMBL22648403

SCHEMBL22648403

CC(C)(C)CC(=O)Nc1cncnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.51
HPGD P15428 3/20 0.51
GAA P10253 1/20 0.51
MAPT P10636 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA14 Q9ULX7 1/20 0.49
NPC1 O15118 2/20 0.47
SMN1; SMN2 Q16637 3/20 0.45
HTT P42858 2/20 0.45
ADORA2A P29274 2/20 0.44
BCAT2 O15382 1/20 0.43
AAK1 Q2M2I8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADORA1 P30542 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19125752 0.82 BCAT2 (0.41) SMN1; SMN2BCAT2
SCHEMBL19169609 0.80 HPGD (0.53) RAB9AHPGDGAAMAPTMEN1
SCHEMBL19169876 0.80 HDAC3 (0.60) RAB9AHPGDGAAMAPTMEN1
SCHEMBL12655416 0.79 SMN1; SMN2 (0.50) RAB9AHPGDGAAMAPTMEN1
SCHEMBL15325536 0.78 HPGD (0.48) RAB9AHPGDGAAMAPTMEN1
SCHEMBL12011608 0.78 HDAC4 (0.48) RAB9AHPGDGAAMAPTMEN1
SCHEMBL23518443 0.78 RAB9A (0.76) RAB9AHPGDGAAMAPTMEN1
SCHEMBL1947815 0.78 HPGD (0.62) RAB9AHPGDGAAMAPTMEN1
SCHEMBL13781504 0.78 RAB9A (0.60) RAB9AHPGDGAAMAPTMEN1
SCHEMBL18836497 0.76 KLK6 (0.39) BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200354367-A1 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200354367-A1 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION XBP1, RNASE1, ERN1 RAB9A 2652/4885HPGD 3731/4885GAA 548/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.