SCHEMBL22650373

SCHEMBL22650373

CC(C)n1cnc2c(F)nc(C(=N)/C(F)=C\N)cc21

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.39
CDK1 P06493 3/20 0.35
CDK2 P24941 3/20 0.35
CCNB1 P14635 2/20 0.35
CCNE1 P24864 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.33
APAF1 O14727 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33
PI4K2A Q9BTU6 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
NPC1 O15118 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650747 0.71 SMN1; SMN2 (0.42) SMN1; SMN2CDK1CDK2CCNB1CCNE1
SCHEMBL22650746 0.69 SMN1; SMN2 (0.45) SMN1; SMN2CDK1CDK2CCNB1CCNE1
SCHEMBL24021324 0.62 CDK4 (0.35) CDK1CDK2CCNB1CCNE1
SCHEMBL22650600 0.61 MAPK14 (0.40) SMN1; SMN2CDK1CDK2L3MBTL1APAF1
SCHEMBL22650364 0.60 CDK4 (0.37) SMN1; SMN2CDK2CDK5CDK5R1
SCHEMBL22650372 0.60 SMN1; SMN2 (0.36) SMN1; SMN2CDK2CDK5CDK5R1
SCHEMBL19397176 0.60 SMN1; SMN2 (0.51) SMN1; SMN2CDK1CDK2CCNB1CCNE1
SCHEMBL20600683 0.59 SMN1; SMN2 (0.46) SMN1; SMN2CDK1CDK2CCNB1CCNE1
SCHEMBL26515108 0.59 SMN1; SMN2 (0.50) SMN1; SMN2CDK1CDK2CCNB1CCNE1
SCHEMBL16938822 0.58 HCAR3 (0.43) SMN1; SMN2CDK2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed