SCHEMBL22650393

SCHEMBL22650393

COc1nc(Cl)cc2c1nc(C)n2C1CCCC1O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
CD274 Q9NZQ7 3/20 0.32
PDCD1 Q15116 2/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RORC P51449 1/20 0.31
PDCD1LG2 Q9BQ51 1/20 0.30
PDE4D Q08499 1/20 0.30
PRPS1 P60891 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29491154 1.00 CCNT1 (0.36) CCNT1CDK9JAK2JAK1CD274
SCHEMBL29491148 0.85 CCNT1 (0.39) CCNT1CDK9JAK2JAK1KDM4E
SCHEMBL22650400 0.85 CCNT1 (0.39) CCNT1CDK9JAK2JAK1KDM4E
SCHEMBL22650391 0.83 JAK2 (0.32) JAK2JAK1
SCHEMBL22650399 0.79 CDK4 (0.33) JAK2JAK1CD274PDCD1RORC
SCHEMBL29491180 0.68 DAPK1 (0.33)
SCHEMBL22650743 0.68 DAPK1 (0.33)
SCHEMBL29491138 0.62 AHCY (0.37)
SCHEMBL9786783 0.59 AHCY (0.50)
SCHEMBL21391183 0.59 CYP11B2 (0.46) CCNT1CDK9KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114364675-A CDK inhibitors 上海齐鲁锐格医药研发有限公司 2022-04-15 CN disclosed
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed