SCHEMBL22650396

SCHEMBL22650396

CC(C)c1cnn2ccc(-c3nc(Nc4ccc(N5CCOCC5=O)c(F)c4)ncc3F)cc12

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 18/20 0.47
CSF1R P07333 17/20 0.47
CDK4 P11802 16/20 0.47
PIK3CD O00329 5/20 0.43
CCNA2 P20248 3/20 0.42
CDK2 P24941 3/20 0.42
CCNE1 P24864 1/20 0.42
JAK2 O60674 2/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41
CCNK O75909 2/20 0.40
CDK7 P50613 2/20 0.40
CDK9 P50750 2/20 0.40
CCNH P51946 2/20 0.40
CDK5 Q00535 2/20 0.40
CDK5R1 Q15078 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650406 0.92 CDK6 (0.44) CDK6CSF1RCDK4PIK3CDCCNA2
SCHEMBL22650401 0.91 NTRK1 (0.46) CDK6CSF1RCDK4CCNA2CDK2
SCHEMBL22650487 0.86 CDK4 (0.42) CDK6CSF1RCDK4PIK3CDCCNA2
SCHEMBL22650591 0.85 CDK6 (0.48) CDK6CSF1RCDK4PIK3CDCCNA2
SCHEMBL22650476 0.79 CDK6 (0.48) CDK6CSF1RCDK4CCNA2CDK2
SCHEMBL22650482 0.76 CDK1 (0.59) CDK6CDK4CCNA2CDK2CCNE1
SCHEMBL22650852 0.76 CDK2 (0.59) CDK6CDK4CCNA2CDK2CCNE1
SCHEMBL22650426 0.76 IKBKB (0.42) CDK6CSF1RCDK4CCNA2CDK2
SCHEMBL22650922 0.76 F10 (0.38) JAK2JAK1TYK2JAK3
SCHEMBL22650475 0.76 CDK6 (0.58) CDK6CSF1RCDK4PIK3CDCCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed