SCHEMBL22650406

SCHEMBL22650406

CC(C)c1cnn2ccc(-c3nc(Nc4ccc(N5CCOCC5=O)c(C(F)(F)F)c4)ncc3F)cc12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 16/20 0.44
CDK4 P11802 14/20 0.44
CSF1R P07333 13/20 0.44
LRRK2 Q5S007 1/20 0.42
PIK3CD O00329 5/20 0.38
CCNA2 P20248 4/20 0.38
CDK2 P24941 4/20 0.38
F10 P00742 2/20 0.38
CCNK O75909 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
CCNH P51946 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
JAK2 O60674 1/20 0.38
CCNE1 P24864 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650396 0.92 CDK6 (0.47) CDK6CDK4CSF1RPIK3CDCCNA2
SCHEMBL22650401 0.88 NTRK1 (0.46) CDK6CDK4CSF1RCCNA2CDK2
SCHEMBL22650487 0.83 CDK4 (0.42) CDK6CDK4CSF1RLRRK2PIK3CD
SCHEMBL22650591 0.82 CDK6 (0.48) CDK6CDK4CSF1RPIK3CDCCNA2
SCHEMBL22650476 0.76 CDK6 (0.48) CDK6CDK4CSF1RCCNA2CDK2
SCHEMBL22650482 0.74 CDK1 (0.59) CDK6CDK4CCNA2CDK2CDK9
SCHEMBL22650852 0.74 CDK2 (0.59) CDK6CDK4CCNA2CDK2CDK7
SCHEMBL22650922 0.73 F10 (0.38) LRRK2F10JAK2
SCHEMBL22650475 0.73 CDK6 (0.58) CDK6CDK4CSF1RPIK3CDCCNA2
SCHEMBL29491147 0.69 CDK6 (0.54) CDK6CDK4CSF1RPIK3CDCCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed