SCHEMBL22650408

SCHEMBL22650408

CN(C(=O)OC(C)(C)C)C1CCCN(c2ccc(N)cn2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.36
RET P07949 2/20 0.36
AAK1 Q2M2I8 1/20 0.36
PDE10A Q9Y233 1/20 0.35
MAP4K4 O95819 2/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
KDM4D Q6B0I6 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
GPR119 Q8TDV5 3/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
HDAC1 Q13547 1/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650381 0.84 ROCK2 (0.38) KDM4DGPR119USP30ROCK2
SCHEMBL22650346 0.81 ROCK2 (0.37) AAK1JAK2JAK1JAK3KDM4D
SCHEMBL15197532 0.79 RET (0.53) PDK2RETAAK1PDE10AMAP4K4
SCHEMBL595584 0.78 AAK1 (0.47) PDK2RETAAK1PDE10AMAP4K4
SCHEMBL22650386 0.78 MAP4K4 (0.44) PDE10AMAP4K4JAK3DDB1CRBN
SCHEMBL529747 0.77 AAK1 (0.54) PDK2RETAAK1PDE10AMAP4K4
SCHEMBL2236554 0.77 AAK1 (0.54) PDK2RETAAK1PDE10AMAP4K4
SCHEMBL12265185 0.77 AAK1 (0.54) PDK2RETAAK1PDE10AMAP4K4
SCHEMBL29418458 0.76 KDM4D (0.38) KDM4DGPR119
SCHEMBL30599761 0.76 KDM4D (0.38) KDM4DGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed