SCHEMBL22650346

SCHEMBL22650346

CN(C(=O)OC(C)(C)C)C1CCCN(c2ccc(N)nc2)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.37
GCK P35557 1/20 0.34
GCKR Q14397 1/20 0.34
GPR119 Q8TDV5 1/20 0.34
ALOX5AP P20292 4/20 0.33
FEN1 P39748 4/20 0.33
LIPE Q05469 2/20 0.33
SPR P35270 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
MMP1 P03956 1/20 0.33
KDM4D Q6B0I6 1/20 0.33
CDK4 P11802 3/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650381 0.86 ROCK2 (0.38) ROCK2GPR119LIPEMMP1KDM4D
SCHEMBL22650408 0.81 PDK2 (0.36) ROCK2GPR119JAK2JAK1JAK3
SCHEMBL22650588 0.81 AKR1C3 (0.36) ROCK2GCKGCKRCDK4PIK3CA
SCHEMBL22650383 0.80 FPR2 (0.35) ROCK2LIPEKDM4DHTR2AHTR2C
SCHEMBL23104497 0.80 RET (0.45) ALOX5APFEN1SPRJAK2JAK1
SCHEMBL29736351 0.80 RET (0.45) ALOX5APFEN1SPRJAK2JAK1
SCHEMBL29491165 0.80 SPR (0.38) ROCK2GPR119SPRJAK2JAK1
SCHEMBL23104405 0.80 RET (0.45) ALOX5APFEN1SPRJAK2JAK1
SCHEMBL22650412 0.80 SPR (0.38) ROCK2GPR119SPRJAK2JAK1
SCHEMBL30700827 0.78 AAK1 (0.43) GCKGCKRGPR119JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed