SCHEMBL22650381

SCHEMBL22650381

CN(C(=O)OC(C)(C)C)C1CCCN(c2ccc(N)cc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.38
LIPE Q05469 2/20 0.37
HRH3 Q9Y5N1 2/20 0.35
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
GPR119 Q8TDV5 4/20 0.34
FPR1 P21462 2/20 0.34
FPR2 P25090 2/20 0.34
KDM4D Q6B0I6 1/20 0.33
NR1H2 P55055 1/20 0.33
MMP1 P03956 1/20 0.33
F10 P00742 2/20 0.33
USP30 Q70CQ3 1/20 0.32
HSD11B1 P28845 1/20 0.32
CASP6 P55212 1/20 0.32
GFER P55789 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650346 0.86 ROCK2 (0.37) ROCK2LIPEGPR119KDM4DMMP1
SCHEMBL22650383 0.85 FPR2 (0.35) ROCK2LIPEHRH3FPR1FPR2
SCHEMBL22650408 0.84 PDK2 (0.36) ROCK2GPR119KDM4DUSP30
SCHEMBL23975899 0.82 RIPK1 (0.42)
SCHEMBL22650413 0.78 DDB1 (0.38) ROCK2HDAC8HDAC6FPR1FPR2
SCHEMBL5958870 0.78 HDAC8 (0.37) HDAC8HDAC6FPR1FPR2F10
SCHEMBL30599761 0.76 KDM4D (0.38) GPR119KDM4D
SCHEMBL29418458 0.76 KDM4D (0.38) GPR119KDM4D
SCHEMBL594199 0.76 GPR119 (0.46) GPR119KDM4DUSP30HSD11B1CASP6
SCHEMBL14022306 0.75 FPR2 (0.45) FPR1FPR2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed