SCHEMBL22650781

SCHEMBL22650781

CC(C)n1cnc2c(F)nc(-c3ccnc(Nc4ccc(N5CCC(N(C)C)CC5=O)cc4)n3)cc21

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
IKBKG Q9Y6K9 1/20 0.39
SYK P43405 2/20 0.36
EGFR P00533 2/20 0.35
WEE1 P30291 4/20 0.35
CDK2 P24941 8/20 0.34
CCNA2 P20248 3/20 0.34
CCNA1 P78396 3/20 0.34
CDK4 P11802 2/20 0.34
CCND1 P24385 2/20 0.34
CDK1 P06493 2/20 0.34
GSK3B P49841 1/20 0.34
KCNH2 Q12809 2/20 0.33
MAPK1 P28482 1/20 0.33
MAP2K1 Q02750 1/20 0.33
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
CCNB1 P14635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650574 0.91 CDK4 (0.43) CDK2CCNA2CCNA1CDK4CCND1
SCHEMBL22650541 0.91 EGFR (0.36) IKBKBCHUKIKBKGSYKEGFR
SCHEMBL22650631 0.89 EGFR (0.43) EGFRCDK2
SCHEMBL22650578 0.88 IKBKB (0.35) IKBKBCHUKIKBKGEGFRCDK2
SCHEMBL22650625 0.87 EGFR (0.43) EGFRCDK2CDK4CCND1CDK1
SCHEMBL22650536 0.85 JAK2 (0.34) IKBKBCHUKIKBKGSYKEGFR
SCHEMBL22650630 0.82 CDK9 (0.35) EGFRCDK2CCNA2CCNA1CDK1
SCHEMBL22650620 0.82 CDK2 (0.36) SYKEGFRCDK2CCNA2CCNA1
SCHEMBL22650626 0.81 CDK2 (0.39) SYKWEE1CDK2CCNA2CCNA1
SCHEMBL22650777 0.81 ACVR1 (0.35) SYKEGFRWEE1CDK2CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed