SCHEMBL22650427

SCHEMBL22650427

CNC1CCCN(c2ccc(Nc3nccc(-c4ccn5ncc(C(C)C)c5c4)n3)c(F)c2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.36
CDK4 P11802 3/20 0.35
CCND3 P30281 3/20 0.35
CDK6 Q00534 3/20 0.35
BTK Q06187 4/20 0.33
MAPK3 P27361 3/20 0.33
MAPK1 P28482 3/20 0.33
ROCK2 O75116 3/20 0.33
INSR P06213 2/20 0.32
IGF1R P08069 1/20 0.32
CDK1 P06493 1/20 0.32
CCNA2 P20248 1/20 0.32
FPR2 P25090 1/20 0.32
CDK9 P50750 1/20 0.32
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650519 0.91 EGFR (0.36) EGFRCDK4CCND3CDK6MAPK3
SCHEMBL22650707 0.90 JAK2 (0.39) CDK4BTKROCK2CDK1CDK9
SCHEMBL22650450 0.88 CDK4 (0.41) CDK4CCND3CDK6CDK1CCNA2
SCHEMBL22650940 0.83 BTK (0.38) CDK4BTKCDK1CDK9
SCHEMBL22650597 0.82 EGFR (0.37) EGFRCDK4MAPK3MAPK1CCNA2
SCHEMBL22650922 0.82 F10 (0.38) EGFRJAK2JAK3
SCHEMBL22650524 0.82 CDK6 (0.38) EGFRCDK4CCND3CDK6MAPK3
SCHEMBL22650523 0.82 EGFR (0.42) EGFRIGF1RJAK2
SCHEMBL22650433 0.81 EGFR (0.36) EGFRCDK4CCND3CDK6MAPK3
SCHEMBL22650709 0.81 JAK2 (0.39) CDK4CDK1CDK9JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed