SCHEMBL22650433

SCHEMBL22650433

CCNC1CCN(c2ccc(Nc3nccc(-c4ccn5ncc(C(C)C)c5c4)n3)c(F)c2)C(=O)C1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.36
MAPK1 P28482 9/20 0.35
MAPK3 P27361 8/20 0.35
CDK4 P11802 1/20 0.32
CCND3 P30281 1/20 0.32
CDK6 Q00534 1/20 0.32
IKBKE Q14164 1/20 0.32
TBK1 Q9UHD2 1/20 0.32
MAPK8 P45983 1/20 0.32
PIK3CG P48736 1/20 0.32
GSK3B P49841 1/20 0.32
CAMKK2 Q96RR4 1/20 0.32
ZAP70 P43403 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650457 0.88 CDK4 (0.40) CDK4CCND3CDK6IKBKETBK1
SCHEMBL22650597 0.88 EGFR (0.37) EGFRMAPK1MAPK3CDK4MAPK8
SCHEMBL22650434 0.84 JAK2 (0.36) CDK4
SCHEMBL22650922 0.83 F10 (0.38) EGFRMAPK8
SCHEMBL22650524 0.83 CDK6 (0.38) EGFRMAPK1MAPK3CDK4CCND3
SCHEMBL22650760 0.82 CDK4 (0.39) CDK4CCND3CDK6GSK3B
SCHEMBL22650519 0.82 EGFR (0.36) EGFRMAPK1MAPK3CDK4CCND3
SCHEMBL22650715 0.81 CDK6 (0.35) EGFRMAPK1MAPK3CDK4CCND3
SCHEMBL22650427 0.81 EGFR (0.36) EGFRMAPK1MAPK3CDK4CCND3
SCHEMBL22650837 0.80 CDK4 (0.41) CDK4CCND3CDK6GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed