SCHEMBL22650715

SCHEMBL22650715

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCC(C)(N)CC5=O)cc4F)n3)cc12

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 6/20 0.35
CCND3 P30281 4/20 0.35
EGFR P00533 1/20 0.35
CDK4 P11802 5/20 0.34
CDK1 P06493 2/20 0.34
CCND1 P24385 2/20 0.34
CCNB1 P14635 1/20 0.34
MAPK3 P27361 5/20 0.33
MAPK1 P28482 5/20 0.33
PIK3CG P48736 3/20 0.32
MAPK8 P45983 2/20 0.32
CAMKK2 Q96RR4 2/20 0.32
CCNA2 P20248 1/20 0.32
MAP3K14 Q99558 3/20 0.32
GSK3B P49841 1/20 0.31
JAK2 O60674 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
BTK Q06187 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650455 0.92 PIK3CG (0.35) CDK6CDK4CDK1CCND1CCNB1
SCHEMBL22650766 0.89 JAK2 (0.39) CDK6CDK4CDK1CCND1CCNB1
SCHEMBL22650755 0.89 CDK4 (0.42) CDK6CCND3CDK4CDK1CCND1
SCHEMBL22650524 0.85 CDK6 (0.38) CDK6CCND3EGFRCDK4CDK1
SCHEMBL22650922 0.85 F10 (0.38) EGFRMAPK8MAP3K14JAK2
SCHEMBL22650597 0.82 EGFR (0.37) EGFRCDK4CCND1MAPK3MAPK1
SCHEMBL22650519 0.82 EGFR (0.36) CDK6CCND3EGFRCDK4CDK1
SCHEMBL22650433 0.81 EGFR (0.36) CDK6CCND3EGFRCDK4MAPK3
SCHEMBL22650427 0.80 EGFR (0.36) CDK6CCND3EGFRCDK4CDK1
SCHEMBL22650705 0.77 CDK6 (0.39) CDK6CCND3CDK4CDK1CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed