SCHEMBL22650549

SCHEMBL22650549

COc1nc(-c2ccnc(Nc3ccc(N4CCNCC4=O)nc3)n2)cc2c1ncn2C(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ZAP70 P43403 11/20 0.42
PRKD3 O94806 2/20 0.42
PRKCG P05129 2/20 0.42
PRKCB P05771 2/20 0.42
LCK P06239 2/20 0.42
PRKCA P17252 2/20 0.42
PRKCH P24723 2/20 0.42
PRKCI P41743 2/20 0.42
PRKCE Q02156 2/20 0.42
PRKCQ Q04759 2/20 0.42
PRKCZ Q05513 2/20 0.42
PRKCD Q05655 2/20 0.42
PRKD1 Q15139 2/20 0.42
EGFR P00533 1/20 0.42
MYLK4 Q86YV6 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
STK17A Q9UEE5 1/20 0.37
TBK1 Q9UHD2 1/20 0.37
WEE1 P30291 2/20 0.36
CCNA2 P20248 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650501 0.88 CDK2 (0.40) ZAP70PRKD3PRKCGPRKCBLCK
SCHEMBL22650496 0.83 EGFR (0.38) ZAP70PRKD3PRKCGPRKCBLCK
SCHEMBL22650502 0.78 CDK4 (0.43) CCNA2CDK2CDK1CCNB1CCNT1
SCHEMBL22650579 0.75 CDK4 (0.48) CCNA2CDK2CDK1CCNB1CCNA1
SCHEMBL22650775 0.74 CDK4 (0.44) CCNA2CDK2CDK1CDK9
SCHEMBL22650464 0.74 CDK6 (0.44) EGFRCCNA2CDK2CCNT1CDK9
SCHEMBL22650515 0.73 SYK (0.35) ZAP70PRKCBEGFRCDK2CDK1
SCHEMBL22650430 0.73 MYLK4 (0.43) ZAP70PRKD3PRKCGPRKCBLCK
SCHEMBL22650503 0.70 MAPK14 (0.46) CCNA2CDK2CDK1CCNB1CCNA1
SCHEMBL22650407 0.70 L3MBTL1 (0.37) CCNA2CDK2CDK1CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed