SCHEMBL22650535

SCHEMBL22650535

CNC1CCCN(c2ccc(Nc3ncc(C)c(-c4cc5c(ncn5C(C)C)c(F)n4)n3)cc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.38
JAK2 O60674 9/20 0.36
TYK2 P29597 7/20 0.36
JAK3 P52333 3/20 0.35
AXL P30530 2/20 0.35
JAK1 P23458 1/20 0.35
FLT3 P36888 1/20 0.35
CDK1 P06493 1/20 0.34
CDK4 P11802 4/20 0.34
CCND1 P24385 4/20 0.34
CCND3 P30281 4/20 0.34
CDK6 Q00534 2/20 0.34
KCNH2 Q12809 1/20 0.34
BRD4 O60885 1/20 0.34
CCND2 P30279 2/20 0.34
FPR1 P21462 1/20 0.34
FPR2 P25090 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650540 0.93 CCND1 (0.40) CDK2AXLCDK4CCND1CCND3
SCHEMBL22650620 0.88 CDK2 (0.36) CDK2JAK2JAK3CDK1KCNH2
SCHEMBL22650619 0.81 CDK4 (0.40) CDK2CDK1CDK4CCND1CCND3
SCHEMBL22650630 0.79 CDK9 (0.35) CDK2JAK2JAK3CDK1KCNH2
SCHEMBL22650536 0.78 JAK2 (0.34) CDK2JAK2JAK3CDK1KCNH2
SCHEMBL22650531 0.75 CDK6 (0.42) CDK2CDK1CDK4CCND1CCND3
SCHEMBL22650578 0.74 IKBKB (0.35) CDK2JAK2JAK3CDK1KCNH2
SCHEMBL22650779 0.74 CDK6 (0.42) CDK2CDK1CDK4CCND1CCND3
SCHEMBL22650626 0.73 CDK2 (0.39) CDK2JAK2JAK3FLT3CDK1
SCHEMBL22650360 0.68 SMN1; SMN2 (0.41) CDK2CDK4CCND1CCND3CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed