SCHEMBL22650540

SCHEMBL22650540

CNC1CCCN(c2ccc(Nc3ncc(Cl)c(-c4cc5c(ncn5C(C)C)c(F)n4)n3)cc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCND1 P24385 10/20 0.40
CDK6 Q00534 10/20 0.40
CDK4 P11802 9/20 0.40
CCND3 P30281 9/20 0.40
CDK2 P24941 1/20 0.36
AXL P30530 1/20 0.35
MAPK10 P53779 3/20 0.35
NTRK1 P04629 1/20 0.35
WEE1 P30291 2/20 0.34
MAPK8 P45983 1/20 0.33
MAPK9 P45984 1/20 0.33
EGFR P00533 1/20 0.33
FPR2 P25090 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650535 0.93 CDK2 (0.38) CCND1CDK6CDK4CCND3CDK2
SCHEMBL22650620 0.87 CDK2 (0.36) CDK2EGFR
SCHEMBL22650619 0.80 CDK4 (0.40) CCND1CDK6CDK4CCND3CDK2
SCHEMBL22650630 0.78 CDK9 (0.35) CDK2MAPK10EGFR
SCHEMBL22650536 0.77 JAK2 (0.34) CDK2EGFR
SCHEMBL22650782 0.75 CTSC (0.40) CCND1CDK6CDK4CCND3CDK2
SCHEMBL22650531 0.74 CDK6 (0.42) CCND1CDK6CDK4CCND3CDK2
SCHEMBL22650578 0.73 IKBKB (0.35) CDK2EGFR
SCHEMBL22650626 0.72 CDK2 (0.39) CDK2MAPK10WEE1MAPK8MAPK9
SCHEMBL22650364 0.70 CDK4 (0.37) CCND1CDK6CDK4CCND3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed