SCHEMBL22650541

SCHEMBL22650541

CC(C)n1cnc2c(F)nc(-c3ccnc(Nc4ccc(N5CCC(N(C)C)CC5=O)cc4F)n3)cc21

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.36
CDK4 P11802 3/20 0.33
CCND1 P24385 3/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
CCNA1 P78396 2/20 0.33
GSK3B P49841 1/20 0.33
PLK1 P53350 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
IKBKB O14920 1/20 0.32
CHUK O15111 1/20 0.32
IKBKG Q9Y6K9 1/20 0.32
ALK Q9UM73 3/20 0.32
SYK P43405 2/20 0.31
CCNT1 O60563 1/20 0.31
CDK9 P50750 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650631 0.93 EGFR (0.43) EGFRCDK2PLK1MKNK1MKNK2
SCHEMBL22650781 0.91 IKBKB (0.39) EGFRCDK4CCND1CCNA2CDK2
SCHEMBL22650574 0.89 CDK4 (0.43) CDK4CCND1CCNA2CDK2CCNA1
SCHEMBL22650532 0.83 EGFR (0.36) EGFRCDK4CCND1MKNK1MKNK2
SCHEMBL22650624 0.82 EGFR (0.34) EGFR
SCHEMBL22650858 0.79 CDK4 (0.41) CDK4CCND1CCNA2CDK2CCNA1
SCHEMBL22650578 0.79 IKBKB (0.35) EGFRCCNA2CDK2CCNA1IKBKB
SCHEMBL22650625 0.78 EGFR (0.43) EGFRCDK4CCND1CDK2
SCHEMBL22650779 0.78 CDK6 (0.42) CDK4CCND1CCNA2CDK2CCNA1
SCHEMBL22650597 0.78 EGFR (0.37) EGFRCDK4CCND1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed