SCHEMBL22650532

SCHEMBL22650532

CC(C)n1cnc2c(F)nc(-c3ccnc(Nc4ccc(N5CCCC(N)C5=O)cc4F)n3)cc21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.36
CDK9 P50750 5/20 0.33
CDK4 P11802 3/20 0.33
CCNT1 O60563 1/20 0.33
CCND1 P24385 1/20 0.33
CCND3 P30281 2/20 0.32
CDK6 Q00534 2/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
BRD4 O60885 3/20 0.31
PIM1 P11309 2/20 0.31
PIM3 Q86V86 2/20 0.31
PIM2 Q9P1W9 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650630 0.90 CDK9 (0.35) EGFRCDK9BRD4
SCHEMBL22650541 0.83 EGFR (0.36) EGFRCDK9CDK4CCNT1CCND1
SCHEMBL22650624 0.82 EGFR (0.34) EGFRCCND3CDK6
SCHEMBL22650620 0.81 CDK2 (0.36) EGFRCDK9BRD4
SCHEMBL22650536 0.80 JAK2 (0.34) EGFRCDK9BRD4
SCHEMBL22650619 0.79 CDK4 (0.40) CDK9CDK4CCNT1CCND1CCND3
SCHEMBL22650627 0.78 CDK4 (0.39) CDK9CDK4CCNT1CCND1CCND3
SCHEMBL22650519 0.77 EGFR (0.36) EGFRCDK9CDK4CCND1CCND3
SCHEMBL22650578 0.77 IKBKB (0.35) EGFRCDK9BRD4
SCHEMBL22650626 0.76 CDK2 (0.39) CDK9CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed