SCHEMBL22650631

SCHEMBL22650631

COc1cc(N2CCC(N(C)C)CC2=O)ccc1Nc1nccc(-c2cc3c(ncn3C(C)C)c(F)n2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.43
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
ALK Q9UM73 5/20 0.39
PLK1 P53350 2/20 0.38
TTK P33981 1/20 0.38
ZAP70 P43403 1/20 0.38
IGF1R P08069 3/20 0.38
INSR P06213 2/20 0.38
AURKA O14965 1/20 0.38
ROS1 P08922 1/20 0.38
EML4 Q9HC35 1/20 0.38
DYRK3 O43781 1/20 0.36
CDK2 P24941 1/20 0.36
CLK1 P49759 1/20 0.36
CLK2 P49760 1/20 0.36
CDK5 Q00535 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDK5R1 Q15078 1/20 0.36
DYRK2 Q92630 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650541 0.93 EGFR (0.36) EGFRMKNK1MKNK2ALKPLK1
SCHEMBL22650781 0.89 IKBKB (0.39) EGFRCDK2
SCHEMBL22650574 0.87 CDK4 (0.43) CDK2CDK5CDK5R1
SCHEMBL22650858 0.79 CDK4 (0.41) CDK2CDK5CDK5R1
SCHEMBL22650578 0.78 IKBKB (0.35) EGFRCDK2
SCHEMBL22650625 0.77 EGFR (0.43) EGFRCDK2
SCHEMBL22650779 0.77 CDK6 (0.42) CDK2CDK5CDK5R1
SCHEMBL22650532 0.76 EGFR (0.36) EGFRMKNK1MKNK2
SCHEMBL22650624 0.75 EGFR (0.34) EGFR
SCHEMBL22650536 0.75 JAK2 (0.34) EGFRCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed