SCHEMBL22650624

SCHEMBL22650624

CC(C)n1cnc2c(F)nc(-c3ccnc(Nc4ccc(N5CCC(C)(N)CC5=O)cc4F)n3)cc21

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.34
CCND3 P30281 1/20 0.32
CDK6 Q00534 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650618 0.93 TTK (0.33) EGFRCCND3CDK6
SCHEMBL22650777 0.90 ACVR1 (0.35) EGFRCDK6
SCHEMBL22650576 0.90 CDK6 (0.38) CCND3CDK6
SCHEMBL22650541 0.82 EGFR (0.36) EGFR
SCHEMBL22650532 0.82 EGFR (0.36) EGFRCCND3CDK6
SCHEMBL22650513 0.80 CDK4 (0.36) CCND3CDK6
SCHEMBL22650715 0.77 CDK6 (0.35) EGFRCCND3CDK6
SCHEMBL22650496 0.76 EGFR (0.38) EGFRCCND3CDK6
SCHEMBL22650579 0.76 CDK4 (0.48) CCND3CDK6
SCHEMBL22650875 0.76 TYK2 (0.44) CCND3CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed