SCHEMBL22650908

SCHEMBL22650908

Fc1cnc(Cl)nc1-c1ccn2ncc(C3CCCC3)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMKK1 Q8N5S9 3/20 0.38
CAMKK2 Q96RR4 3/20 0.38
KMT2A Q03164 1/20 0.36
ADH5 P11766 1/20 0.32
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
RPS6KA5 O75582 1/20 0.31
SCN5A Q14524 1/20 0.31
MAPK1 P28482 3/20 0.30
MAPT P10636 1/20 0.30
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
MAPK3 P27361 1/20 0.30
PIK3CA P42336 1/20 0.30
CDK6 Q00534 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30
POLB P06746 1/20 0.30
CASP6 P55212 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650436 0.80 RPS6KA5 (0.34) RPS6KA5SCN5AMAPTPOLBCASP6
SCHEMBL22650356 0.77 SCN5A (0.39) RPS6KA5SCN5A
SCHEMBL22650740 0.77 RPS6KA5 (0.32) CAMKK2RPS6KA5
SCHEMBL22650437 0.72 SCN5A (0.42) RPS6KA5SCN5AMAPTPOLBCASP6
SCHEMBL22650698 0.72 MAPK14 (0.35) MAPK1CDK2PIK3CA
SCHEMBL31334301 0.71 KMT2A (0.38) KMT2AMAPTCCNA2CDK2CDK6
SCHEMBL19966454 0.70 KMT2A (0.40) KMT2ACCNA2CDK2PIK3CACDK6
SCHEMBL28987249 0.70 KMT2A (0.40) KMT2ACDK2PIK3CACDK6
SCHEMBL30278677 0.70 KMT2A (0.40) KMT2ACDK2PIK3CACDK6
SCHEMBL15252527 0.69 CDK9 (0.51) MAPTCDK2CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed