SCHEMBL22650918

SCHEMBL22650918

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(S(N)(=O)=O)cc4)n3)cc12

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DKK1 O94907 2/20 0.57
GSK3B P49841 2/20 0.57
IKBKB O14920 11/20 0.55
MAPK8 P45983 1/20 0.53
MAPK10 P53779 1/20 0.53
CDK2 P24941 3/20 0.51
SMG1 Q96Q15 2/20 0.51
CCNT1 O60563 2/20 0.50
CDK1 P06493 2/20 0.50
CCNB1 P14635 2/20 0.50
CDK9 P50750 2/20 0.50
CCNA2 P20248 1/20 0.50
CDK7 P50613 1/20 0.50
CCNH P51946 1/20 0.50
CCNA1 P78396 1/20 0.50
MTOR P42345 1/20 0.49
IGF1R P08069 1/20 0.48
JAK2 O60674 1/20 0.48
CHUK O15111 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650923 0.85 MAPK8 (0.54) GSK3BIKBKBMAPK8MAPK10CDK2
SCHEMBL22650852 0.84 CDK2 (0.59) IKBKBCDK2CCNT1CDK1CCNB1
SCHEMBL22650920 0.83 CDK2 (0.54) MAPK8MAPK10CDK2CDK1CCNB1
SCHEMBL22650919 0.82 CDK2 (0.54) GSK3BMAPK8MAPK10CDK2CDK1
SCHEMBL22650921 0.80 MTOR (0.49) IKBKBCDK2SMG1CDK1CCNB1
SCHEMBL22650595 0.79 PRKCA (0.40) GSK3BCDK2CCNT1CDK1CCNB1
SCHEMBL22650796 0.78 CDK2 (0.44) IKBKBCDK2SMG1CDK1CCNB1
SCHEMBL22650422 0.78 CDK1 (0.41) CDK2CCNT1CDK1CCNB1CDK9
SCHEMBL22650849 0.78 CDK1 (0.47) IKBKBCDK2SMG1CDK1MTOR
SCHEMBL22650482 0.77 CDK1 (0.59) GSK3BCDK2CCNT1CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed