SCHEMBL2265192

SCHEMBL2265192

Cn1cc(-n2ccc(=O)c(Cc3cccc(N(CC(F)(F)CN4CCOCC4)C(=O)O)c3)n2)cn1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
MCHR1 Q99705 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13275099 0.88 CASR (0.36) HDAC1HDAC8HDAC6MCHR1SMN1; SMN2
SCHEMBL2349823 0.87 ENPP2 (0.32)
SCHEMBL2361416 0.87 ENPP2 (0.34)
SCHEMBL2222897 0.87 SMN1; SMN2 (0.36) HDAC1HDAC8HDAC6MCHR1SMN1; SMN2
SCHEMBL2266173 0.85 HDAC1 (0.32) HDAC1HDAC8HDAC6MCHR1SMN1; SMN2
SCHEMBL13506838 0.84 ENPP2 (0.34)
SCHEMBL2365229 0.83 CCNC (0.34)
SCHEMBL2221295 0.83 BRD4 (0.34)
SCHEMBL2269504 0.82 CREBBP (0.34)
SCHEMBL2221688 0.82 OPRM1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO claimed
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed