SCHEMBL2222897

SCHEMBL2222897

Cn1cc(-n2ccc(=O)c(Cc3cccc(N(CCCN4CCOCC4)C(=O)O)c3)n2)cn1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
PLA2G7 Q13093 1/20 0.35
PARP1 P09874 1/20 0.35
NAMPT P43490 3/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MAPK1 P28482 2/20 0.34
TP53 P04637 1/20 0.34
MAPK14 Q16539 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
CCR5 P51681 2/20 0.34
USP2 O75604 2/20 0.33
TSHR P16473 1/20 0.33
TACR2 P21452 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MCHR1 Q99705 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13275099 0.95 CASR (0.36) SMN1; SMN2L3MBTL1PLA2G7PARP1HDAC1
SCHEMBL2219314 0.92 CCR5 (0.34) PLA2G7PARP1CCR5
SCHEMBL2274437 0.91 CCR5 (0.34) CCR5MCHR1
SCHEMBL2265615 0.90 FGFR1 (0.35) CCR5
SCHEMBL2221167 0.88 CASR (0.35) SMN1; SMN2L3MBTL1PARP1HDAC1HDAC8
SCHEMBL2362780 0.87 OPRM1 (0.36) PARP1MAPK14MCHR1
SCHEMBL13274618 0.87 CASR (0.34) SMN1; SMN2L3MBTL1PARP1HDAC1HDAC8
SCHEMBL13507143 0.87 ENPP2 (0.33)
SCHEMBL2221295 0.87 BRD4 (0.34) MAPK1
SCHEMBL2266173 0.87 HDAC1 (0.32) SMN1; SMN2L3MBTL1HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO claimed
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed