SCHEMBL22658181

SCHEMBL22658181

CCC(=O)c1cc(NC(=O)O)ccn1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.45
ANO1 Q5XXA6 9/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
PRKCI P41743 1/20 0.42
SMARCA2 P51531 1/20 0.41
SMARCA4 P51532 1/20 0.41
SORT1 Q99523 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17942340 0.81 ALDH1A1 (0.44) ARANO1JAK2JAK1TYK2
SCHEMBL28663446 0.81 KDM4E (0.55) ARANO1SMARCA2SMARCA4SORT1
SCHEMBL22670384 0.80 AR (0.48) ARANO1
SCHEMBL23405316 0.79 ANO1 (0.47) ANO1JAK2TYK2SMARCA2SMARCA4
SCHEMBL15880501 0.78 PRKCI (0.62) ARJAK2JAK1TYK2PRKCI
SCHEMBL28292635 0.78 SCN10A (0.44) ARANO1SMARCA2SMARCA4SORT1
SCHEMBL30885027 0.78 UHRF1 (0.43) KDM4EALDH1A1NPC1RAB9A
SCHEMBL2643034 0.78 UHRF1 (0.43) KDM4EALDH1A1NPC1RAB9A
SCHEMBL28294352 0.77 RAF1 (0.43) ARANO1TYK2SMARCA2SMARCA4
SCHEMBL15880685 0.75 SMARCA2 (0.65) SMARCA2SMARCA4SORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3983386-A1 ACSS2 INHIBITORS AND METHODS OF USE THEREOF Metabomed Ltd (IL) 2022-04-20 EP disclosed
WO-2020230136-A1 ACSS2 INHIBITORS AND METHODS OF USE THEREOF METABOMED LTD (IL) 2020-11-19 WO disclosed