SCHEMBL28294352

SCHEMBL28294352

CN(C)C(=O)c1cc(NC(=O)O)ccn1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 3/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PIK3C3 Q8NEB9 4/20 0.41
SMARCA2 P51531 1/20 0.41
SMARCA4 P51532 1/20 0.41
ANO1 Q5XXA6 3/20 0.40
SORT1 Q99523 2/20 0.40
TYK2 P29597 1/20 0.39
AR P10275 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL883725 0.83 PIK3C3 (0.41) RAF1ALDH1A1KDM4EPIK3C3TYK2
SCHEMBL17942340 0.81 ALDH1A1 (0.44) ALDH1A1KDM4ESMARCA2SMARCA4ANO1
SCHEMBL28663446 0.81 KDM4E (0.55) ALDH1A1KDM4ESMARCA2SMARCA4ANO1
SCHEMBL2437319 0.79 ALDH1A1 (0.41) RAF1ALDH1A1KDM4EPIK3C3ANO1
SCHEMBL2437324 0.79 ALDH1A1 (0.38) RAF1ALDH1A1KDM4EPIK3C3TYK2
SCHEMBL23405316 0.79 ANO1 (0.47) RAF1SMARCA2SMARCA4ANO1SORT1
SCHEMBL28292635 0.78 SCN10A (0.44) RAF1ALDH1A1KDM4ESMARCA2SMARCA4
SCHEMBL4947098 0.78 ALDH1A1 (0.44) RAF1ALDH1A1KDM4EPIK3C3MAPT
SCHEMBL22658181 0.77 AR (0.45) ALDH1A1KDM4ESMARCA2SMARCA4ANO1
SCHEMBL5700562 0.76 ALDH1A1 (0.43) RAF1ALDH1A1KDM4EPIK3C3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed