SCHEMBL28292635

SCHEMBL28292635

NC(=O)c1cc(NC(=O)O)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 8/20 0.44
SMARCA2 P51531 2/20 0.41
SMARCA4 P51532 2/20 0.41
RAF1 P04049 1/20 0.40
ANO1 Q5XXA6 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
TSHR P16473 1/20 0.40
MC4R P32245 1/20 0.40
ADRA1A P35348 1/20 0.40
MC3R P41968 1/20 0.40
GSK3B P49841 2/20 0.40
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
KDR P35968 1/20 0.40
SORT1 Q99523 1/20 0.39
KDM4E B2RXH2 1/20 0.39
KDM6B O15054 1/20 0.39
TET3 O43151 1/20 0.39
KDM4A O75164 1/20 0.39
BBOX1 O75936 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28663446 0.85 KDM4E (0.55) SCN10ASMARCA2SMARCA4ANO1KCNK3
SCHEMBL23488366 0.82 KCNK3 (0.62) KCNK3KCNK9MAPT
SCHEMBL17942340 0.82 ALDH1A1 (0.44) SMARCA2SMARCA4ANO1KCNK3KCNK9
SCHEMBL17076844 0.80 APP (0.43) SCN10ARAF1ADORA3TSHRMC4R
SCHEMBL31633789 0.79 ACVRL1 (0.52) TSHRGSK3BKDRKDM4EALDH1A1
SCHEMBL23405316 0.79 ANO1 (0.47) SMARCA2SMARCA4RAF1ANO1ADORA3
SCHEMBL5007785 0.79 EGFR (0.41) SCN10AANO1KCNK3KCNK9KDR
SCHEMBL22658181 0.78 AR (0.45) SMARCA2SMARCA4ANO1SORT1KDM4E
SCHEMBL28294352 0.78 RAF1 (0.43) SMARCA2SMARCA4RAF1ANO1SORT1
SCHEMBL20652765 0.77 ADORA3 (0.39) SCN10ARAF1ADORA3TSHRMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed