SCHEMBL22685247

SCHEMBL22685247

COc1ccc(C(=O)NC2(c3ccc(-c4cnc(C(F)(F)F)cc4N)cc3)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41
HDAC6 Q9UBN7 3/20 0.40
PTPN1 P18031 1/20 0.40
MAP4K4 O95819 1/20 0.39
CHEK2 O96017 1/20 0.39
HDAC3 O15379 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
DEGS1 O15121 1/20 0.38
F10 P00742 2/20 0.38
POLB P06746 1/20 0.38
PDE2A O00408 3/20 0.38
TSHR P16473 1/20 0.37
IDO1 P14902 2/20 0.37
PTPN11 Q06124 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22685075 0.92 IDO1 (0.43) HDAC6PTPN1MAP4K4CHEK2HDAC3
SCHEMBL22685250 0.91 PTPN1 (0.40) ROCK2ROCK1HDAC6PTPN1HDAC3
SCHEMBL22685264 0.89 PDE2A (0.42) ROCK2ROCK1HDAC6MAP4K4CHEK2
SCHEMBL22685245 0.85 MAP4K4 (0.41) MAP4K4DEGS1PDE2AIDO1CYP2C9
SCHEMBL22685329 0.82 IDO1 (0.43) ROCK2ROCK1HDAC6MAP4K4HDAC3
SCHEMBL22685074 0.80 IDO1 (0.51) HDAC6MAP4K4HDAC3HDAC1HDAC2
SCHEMBL22685249 0.80 WDR91 (0.41) ROCK2ROCK1HDAC6MAP4K4HDAC3
SCHEMBL22685078 0.80 WDR91 (0.53) MAP4K4F10PDE2AIDO1CYP2C9
SCHEMBL22685072 0.80 IDO1 (0.43) HDAC6HDAC3HDAC1HDAC2PDE2A
SCHEMBL22685187 0.79 PDE2A (0.44) ROCK2ROCK1HDAC6HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020228823-A1 NOVEL AMIDE COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2020-11-19 WO disclosed