SCHEMBL22700396

SCHEMBL22700396

COc1ccc(COC[C@H]2OC3CCC(COC(=O)c4ccccc4)(C2O[Si](C)(C)C(C)(C)C)[C@H]3n2cnc3c(Cl)nc(Cl)nc32)cc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.36
NT5E P21589 10/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
BCHE P06276 1/20 0.32
TBXAS1 P24557 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19979255 0.87 PDE2A (0.37) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19979256 0.85 NT5E (0.39) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19975506 0.85 NT5E (0.39) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19979002 0.81 PDE2A (0.33) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19975504 0.76 NT5E (0.39) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19979067 0.74 LMNA (0.40) NT5EALDH1A1LMNATP53MAPT
SCHEMBL19974569 0.72 ADORA2A (0.41) NT5EALDH1A1LMNATP53MAPT
SCHEMBL19974567 0.71 TBXAS1 (0.37) NT5EALDH1A1MAPTTDP1TBXAS1
SCHEMBL22700325 0.70 LMNA (0.42) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19974597 0.69 NT5E (0.36) NT5ETDP1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512860-B1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC (CA) 2020-11-25 EP disclosed