SCHEMBL19979002

SCHEMBL19979002

COc1ccc(COC[C@H]2OC3[C@@H]4C(COC(=O)c5ccccc5)(C2O[Si](C)(C)C(C)(C)C)C34n2cnc3c(Cl)nc(Cl)nc32)cc1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.33
TBXAS1 P24557 1/20 0.32
NT5E P21589 2/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
BCHE P06276 1/20 0.31
HRAS P01112 1/20 0.30
DHODH Q02127 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19979255 0.86 PDE2A (0.37) PDE2ATBXAS1NT5EALDH1A1LMNA
SCHEMBL19975506 0.84 NT5E (0.39) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19979256 0.84 NT5E (0.39) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL22700396 0.81 PDE2A (0.36) PDE2ATBXAS1NT5EALDH1A1LMNA
SCHEMBL19979098 0.80 LMNA (0.37) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19975504 0.74 NT5E (0.39) PDE2ANT5EALDH1A1LMNATP53
SCHEMBL19974567 0.73 TBXAS1 (0.37) TBXAS1NT5EALDH1A1MAPTTDP1
SCHEMBL19979067 0.71 LMNA (0.40) NT5EALDH1A1LMNATP53MAPT
SCHEMBL19974597 0.71 NT5E (0.36) TBXAS1NT5ETDP1DHODH
SCHEMBL22700167 0.70 TBXAS1 (0.35) TBXAS1NT5EDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049534-A1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC. (CA) 2018-03-22 WO disclosed